Biosynthesis of Polyphenols with Antioxidant Potential: A Review

Hilda Vasanthakaalam

College of Agriculture, Forestry and Food Science, University of Rwanda, P.O. Box: 210, Musanze, Rwanda.

Justin N. Kabera *

Chemistry Division Manager, Rwanda Forensic Institute, P.O. Box: 979, Kigali, Rwanda.

Vedaste Ndungutse

College of Agriculture, Forestry and Food Science, University of Rwanda, P.O. Box: 210, Musanze, Rwanda.

Jean Paul Hategekimana

College of Agriculture, Forestry and Food Science, University of Rwanda, P.O. Box: 210, Musanze, Rwanda.

*Author to whom correspondence should be addressed.


Abstract

Polyphenols are diverse plant secondary metabolites characterised by phenolic structural units and widely recognised for their antioxidant potential. This chapter reviews the major classes of polyphenols, their biosynthetic origins, biological properties, production approaches, extraction methods, and selected industrial applications. The discussion covers phenolic acids, flavonoids, stilbenes, lignans, tannins, and related compounds, with emphasis on their occurrence in fruits, vegetables, seeds, cereals, nuts, tea, coffee, wine, and other plant-derived materials. It also summarises the shikimate and phenylpropanoid pathways, which contribute to the formation of flavonoids, lignin-related compounds, and other phenolic metabolites. The antioxidant mechanisms described include free-radical scavenging, modulation of oxidative stress, metal-ion interaction, and support of cellular protective systems. Health-related sections outline reported anti-inflammatory, antimicrobial, cardioprotective, antidiabetic, neuroprotective, and anticancer activities, while recognising the need for further validation of mechanisms and effects. The chapter also reviews plant tissue culture, genetic engineering, enzymatic extraction, and fermentation as approaches for controlled production, scalability, and improved recovery of polyphenols. In addition, it outlines applications in food preservation, pharmaceuticals, cosmetics, textiles, paper, and chromatographic identification. Overall, polyphenols are presented as scientifically relevant natural compounds with broad biological and industrial interest, although their practical use depends on validated health claims, production efficiency, product quality, analytical reliability, safety, and reproducibility.

Keywords: Polyphenols, antioxidant potential, phenylpropanoid pathway, shikimate pathway, flavonoids, phenolic acids, plant tissue culture, enzymatic extraction, fermentation, industrial applications


How to Cite

Vasanthakaalam, H., Kabera, J. N., Ndungutse, V., & Hategekimana, J. P. (2026). Biosynthesis of Polyphenols with Antioxidant Potential: A Review. Chemistry and Biochemistry: Research Progress Vol. 11, 152–174. https://doi.org/10.9734/bpi/cbrp/v11/7741